Bhandi neMugwagwa: Kushandira Pamwe, Kuwirirana uye Kukunda-Kukunda
zvigadzirwa

Zvigadzirwa

Empagliflozin CAS:864070-44-0 Mugadziri wezvigadzirwa

Empagliflozin imusanganiswa weC-glycosyl une beta-glucosyl residue ine (4-chloro-3-{4-[(3S)-tetrahydrofuran-3-yloxy]benzyl}phenyl group panzvimbo yeanomeric. Mushonga we sodium-glucose co-transporter 2 unoshandiswa sechibatsiro chekudya uye kurovedza muviri kuvandudza kudzora glycemic muvanhu vakuru vane chirwere cheshuga cherudzi rwechipiri. Unoshanda semushonga we sodium-glucose transport protein subtype 2 uye mushonga we hypoglycemic. Imushonga weC-glycosyl, aromatic ether, tetrahydrofuryl ether uye nhengo ye monochlorobenzenes.


Ruzivo rweChigadzirwa

Matagi eChigadzirwa

Kushandiswa uye Mhedzisiro

Empagliflozin mushonga mutsva, une simba uye unosarudza weSGLT-2 inhibitor, unovandudza kudzora kweglucose uye hunhu hwe metabolic syndrome mumakonzo ane chirwere cheshuga.Empagliflozin (zita rekutengeserana rekuti Jardiance) inhibitor ye sodium glucose co-transporter-2 (SGLT-2), uye inoita kuti shuga muropa ibudiswe neitsvo uye ibviswe muweti.Empagliflozin inogona kukonzera kushaya mvura mumuviri uye kutungamira kudzikira kweBP, zvichikonzera varwere vane dzungu kana kupera simba uye kudzikira kwekushanda kweitsvo. Njodzi yevarwere vakwegura, kunyanya avo vane dambudziko rekushanda kweitsvo uye diuretics, inoita kunge yakakura.FDA inoda kuti Boehring naEli Lilly vaite zvidzidzo zvina zvepashure pekushambadza: miedzo yakazara yemhedzisiro yemwoyo inoenderera mberi, miedzo ye pharmacokinetics yevana uye pharmacodynamics, miedzo yekuchengetedza vana uye kushanda zvakanaka, bvunzo yechepfu yemushonga (kunyanya mhedzisiro yekushanda kweitsvo, mapfupa nekukura nekukura).

Muenzaniso weChigadzirwa

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Kurongedza Chigadzirwa:

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Mamwe Mashoko:

Kuumbwa C23H27ClO7
Kuyedza 99%
Chitarisiko Upfu chena
Nhamba yeCAS 864070-44-0
Kurongedza 25KG
Hupenyu hweSherufu makore maviri
Kuchengetera Chengeta munzvimbo inotonhorera uye yakaoma
Chitupa ISO.

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