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3,3-Dimethyl-1-Butyne CAS:917-92-0
3,3-Dimethyl-1-butyne ikemikari inozivikanwa nechimiro chayo che "triple bond" uye mapoka maviri e "methyl" akabatana nemaatomu ekabhoni e "triple bond". Inowanzonzi tetramethylethyne uye inoshandiswa mumaitiro akasiyana-siyana ekugadzira makemikari.
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6-Chloro-3-methyluracil CAS:4318-56-3
6-Chloro-3-methyluracil inobva kuuracil, pyrimidine base, ine chlorine ne methyl groups zvakabatana nenzvimbo dzakatarwa pauracil ring. Kugadziriswa uku kunopa hunhu hwakasiyana hwemakemikari nehupenyu kune chinhu ichi, zvichiita kuti chive chakakosha mukurapa chemistry uye biochemical research. Maumbirwo e6-Chloro-3-methyluracil anokanganisa kudyidzana kwayo mukati memaitiro ehupenyu, kunyanya mukugadzirwa kwe nucleic acid uye kudzivirira enzyme, izvo zvinhu zvakakosha mukugadzirwa kwemishonga nekukura kwekurapa.
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4-Isothiocyanato-2-(trifluoromethyl)benzonitrile CAS:143782-23-4
4-Isothiocyanato-2- (trifluoromethyl)benzonitrile ikemikari inoonekwa neboka rinoshanda reisothiocyanate rakabatana nerin'i yebenzene yakatsiviwa netrifluoromethyl. Inoshandiswa zvakanyanya sechivako chinoshanda zvakasiyana-siyana mukugadzirwa kwezvinhu zvakasikwa, zvichigonesa kugadzirwa kwemaumbirwo akaomarara emamorekuru nezvinhu zvinoshanda.
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Kubuda(1R,3R)-1-(1,3-Benzodioxol-5-yl)-2-(chloroacetyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylicacidmethyste CAS:171489-59-1
(1R,3R)-1-(1,3-Benzodioxol-5-yl)-2-(chloroacetyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indole-3-carboxylic Acid Methyl Ester, yakapfupikiswa kuti ijekeswe, ikemikari inozivikanwa nekugadzirwa kwayo kwakaoma kwemamorekuru uye mashandisirwo ayo mumishonga. Iyi kemikari inobatanidza pyridoindole core ne tetrahydrofuran ring yakabatana ne chloroacetyl group uye 1,3-benzodioxol-5-yl moiety, ine methyl ester functionality. Izvi zvinhu zvemaumbirwo zvinopa nzira dzekugadzirisa maumbirwo akasiyana-siyana uye kuferefeta kwakazara kwehupenyu.
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Candesartan ester yepakati C3 CAS:136285-65-9
Candesartan ester intermediate C3 chinhu chakakosha mukugadzirwa kweCandesartan cilexetil, mushonga unozivikanwa we angiotensin II receptor antagonist unoshandiswa zvakanyanya kurapa BP uye kusagadzikana kwemoyo. Mushonga uyu une basa rakakosha muindasitiri yemishonga nekuda kwebasa rawo senzira yekutanga mukugadzirwa kweCandesartan cilexetil zvinobudirira.
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Linagliptin interMediate F CAS:853029-57-9
Linagliptin Intermediate F mushonga unobatsira zvikuru mukugadzirwa kwelinagliptin, mushonga une simba we dipeptidyl peptidase-4 (DPP-4) unoshandiswa mukurapa chirwere cheshuga cherudzi rwechipiri. Mushonga uyu une basa guru muindasitiri yemishonga nekuda kwemaumbirwo nemashandiro awo chaiwo emakemikari. Linagliptin, inozivikanwa se (R)-8-(3-aminopiperidin-1-yl)-7-(but-2-yn-1-yl)-3-methyl-1-(2,4,5-trifluorophenyl)-1,2-dihydroquinazolin-2(3H)-one, unoshanda pakurapa nekudzivisa DPP-4 enzyme activity, nokudaro uchisimudzira huwandu hweincretin hormones seGLP-1 (glucagon-like peptide-1). Izvi zvinoita kuti glycemic control ive nani muvarwere vane chirwere cheshuga.
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Candesartan Cilexetil Impurity 8 CAS:139481-28-0
Candesartan Cilexetil Impurity 8 chinhu chinobva pakugadzirwa kweCandesartan cilexetil, mushonga unodzivirira angiotensin II receptor unoshandiswa zvakanyanya kudzora BP nekushaya simba kwemoyo. Kunyangwe usingadiwi mukugadzirwa kwemishonga kwekupedzisira, kunzwisisa nekudzora kusvibiswa kwakakosha pakuona kuchengetedzeka kwechigadzirwa, kushanda zvakanaka, uye kutevedzera mitemo.
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BENZOIC ACID, 2-[[(1,1-DIMETHYLETHOXY)CARBONYL]AMINO]-3-NITRO-METHYL ESTER CAS:57113-90-3
BENZOIC ACID, 2-[[(1,1-DIMETHYLETHOXY)CARBONYL]AMINO]-3-NITRO-METHYL ESTER ikemikari inozivikanwa nekuumbwa kwayo kwakaomarara kwemamorekuru uye kushandiswa kwayo mune zvemishonga. Iyi kemikari inobatanidza benzoic acid core nechikamu checarbamate chine dimethylethoxy group uye nitro-methyl ester functionality, zvichiita kuti ive yakakosha mukurapa chemistry uye biochemical research nekuda kwehunhu hwayo hwakasiyana uye mabasa ayo ehupenyu.
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pyridine-3-sulfonyl chloride CAS:16133-25-8
Pyridine-3-sulfonyl chloride ikemikari inozivikanwa nekushandiswa kwayo kwakasiyana-siyana mukugadzira organic uye kutsvagurudza mishonga. Kemikari iyi, inonziwo picolinoyl chloride, ine pyridine core inotsiviwa neboka resulfonyl chloride panzvimbo ye3, zvichiita kuti ive yakakosha nekuda kwekuita kwayo kwakasiyana uye kugona kwayo kushandiswa mumakemikari akasiyana-siyana.
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5-(2-fluorophenyl)-1H-pyrrole-3-carbonitrile CAS:1240948-77-9
5-(2-Fluorophenyl)-1H-pyrrole-3-carbonitrile ikemikari inosiyaniswa nechimiro chayo chemamorekuru uye mashandisirwo ayo mumakemikari ekurapa uye kugadzirwa kweorganic. Iyi kemikari ine pyrrole core inotsiviwa neboka refluorophenyl neboka recyano panzvimbo dzakatarwa, zvichiita kuti ive yakakosha nekuda kwekusiyana kwayo uye mabasa ayo ehupenyu.
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Vonoprazan CAS:881681-00-1
Vonoprazan imushonga unozivikanwa nekugona kwayo kudzvinyirira acid yemudumbu, zvichiisiyanisa neproton pump inhibitors (PPIs) nekuda kwekushanda kwayo kwakasiyana. Mushonga uyu unodzivisa H+, K+-ATPase proton pump mumasero emudumbu zvine hungwaru uye kushanda zvakanaka, zvichiita kuti acid irambe iripo uye isingaperi.
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N-(4-CYANO-PHENYL)-GLYCINE CAS:42288-26-6
N-(4-Cyano-phenyl)-glycine ikemikari inoratidzwa nechimiro chayo chemamorekuru uye mashandisirwo ayo muzvikamu zvakasiyana-siyana, kunyanya mumakemikari ekurapa uye tsvakurudzo yemakemikari. Iyi kemikari inobatanidza boka rephenyl nechikamu cheglycine, zvichiita kuti ive yakakosha nekuda kwekusiyana kwemaumbirwo ayo uye mabasa ayo ehupenyu.
