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Tetracycline CAS: 60-54-8
Tetracycline mushonga unorwisa mabhakitiriya une spectrum yakakura uri muboka retetracycline, unobva mu chlortetracycline yemusikirwo. Unodzivirira kugadzirwa kwemapuroteni emabhakitiriya nekusungana ne bacterial ribosome, nokudaro uchidzivirira kubatana kwe aminoacyl-tRNA kune mRNA-ribosome complex. Maitiro aya anoita kuti pave nemhedzisiro ye bacteriostatic kurwisa mabhakitiriya akasiyana-siyana e gram-positive ne gram-negative, pamwe nemamwe ma protozoa.
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Teicoplanin CAS:61036-62-2
Teicoplanin mushonga unorwisa mabhakitiriya unobva kuActinoplanes teichomyceticus, unoshanda pakurwisa mabhakitiriya akasiyana-siyana ane gram-positive anosanganisira methicillin-resistant Staphylococcus aureus (MRSA). Unodzivirira kugadzirwa kwemadziro emasero ebhakitiriya nekusunga kune D-alanyl-D-alanine terminus yepeptidoglycan precursors, zvichikonzera lysis yemasero uye mhedzisiro yekuuraya mabhakitiriya. Teicoplanin inowanzoshandiswa muzvipatara kurapa hutachiona hwakasimba hunokonzerwa nezvipembenene zvine gram-positive.
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Sulfisoxazol (4-amino-N-(3,4-dimethyl-5-isoxazolyl)benzenesulfonamide) CAS:127-69-5
Sulfisoxazole, inozivikanwawo sesulfafurazole, mushonga unorwisa mabhakitiriya wesulfonamide uri muboka remishonga yesulfa. Sulfisoxazole, inotsanangurwa se4-amino-N-(3,4-dimethyl-5-isoxazolyl)benzenesulfonamide, inodzivirira kukura kwemabhakitiriya nekuvhiringidza kugadzirwa kwefolic acid. Maitiro aya anotarisa dihydropteroate synthase, enzyme inokosha pakugadzirwa kwebhakitiriya, nokudaro ichidzivisa kukura kwavo nekuwanda kwavo.
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Sulfapyridine CAS:144-83-2
Sulfapyridine mushonga unorwisa mabhakitiriya we sulfonamide waimboshandiswa kare mukurapa hutachiona hwemabhakitiriya, kunyanya munguva yeHondo Yenyika II. Iri muboka remishonga ye sulfa, iyo inodzivirira kukura kwebhakitiriya nekuvhiringidza kugadzirwa kwe folic acid. Sulfapyridine ine simba rayo re bacteriostatic nekutsvaga dihydropteroate synthase, enzyme inokosha pakugadzirwa kwe folate mumabhakitiriya.
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Tazobactam CAS:89786-04-9
Tazobactam mushonga unodzivirira beta-lactamase unowedzera kushanda kwemishonga inorwisa mabhakitiriya yebeta-lactam nekudzivirira kubva mukukuvadzwa nema enzymes ebeta-lactamase anokonzerwa nemabhakitiriya akawanda anodzivirira mabhakitiriya. Inowanzoshandiswa pamwe chete nemishonga inorwisa mabhakitiriya yebeta-lactam yakadai sepiperacillin kuwedzera kushanda kwayo mukurwisa hutachiona hwakasiyana-siyana hwemabhakitiriya. Tazobactam inonyatso dzorera kushanda kwemishonga inorwisa mabhakitiriya yebeta-lactam mukurwisa mabhakitiriya anogadzira beta-lactamase, kunyanya zvipembenene zvisina gram.
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Tigecycline CAS:220620-09-7
Tigecycline mushonga unorwisa mabhakitiriya weglycylcycline une spectrum yakakura unodzivirira kugadzirwa kwemapuroteni emabhakitiriya nekusunga ku30S ribosomal subunit, nokudaro uchiita kuti pave nemigumisiro yebhakitiriya pakurwisa mabhakitiriya akasiyana-siyana ane gram-positive negram-negative, kusanganisira mabhakitiriya asingapindi mishonga yakawanda. Muchimiro chayo wakabatana netetracyclines asi une simba rakawanda pakurwisa mabhakitiriya asingapindi mishonga nekuda kwekushanda kwayo kwakasiyana uye kugadziriswa kwechimiro.
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Sulbactam sodium munyu CAS:69388-84-7
Munyu weSulbactam sodium inhibitor ye beta-lactamase inowanzoshandiswa pamwe chete nemamwe maantibiotics kurwisa hutachiona hwebhakitiriya. Inoshanda nekudzivisa mashandiro ema enzymes e beta-lactamase anogadzirwa nemabhakitiriya, izvo zvinogona kuita kuti maantibiotic asashande. Nekudzivirira kuparara kwemishonga inorwisa mabhakitiriya yakaita sepenicillins ne cephalosporins, munyu we sulbactam sodium unobatsira kuwedzera hunhu hwavo hwemaantibacterial. Mushonga uyu unowanzo shandiswa pamwe chete nemishonga inorwisa mabhakitiriya yakaita se ampicillin kugadzira mhedzisiro inoshanda kurwisa mhando dzakasiyana dzebhakitiriya dzinokurumidza kubatwa.
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Sulfadimidine CAS:57-68-1
Sulfadimidine, inozivikanwawo sesulfamethazine, mushonga unorwisa mabhakitiriya unoshandiswa mukurapa hutachiona hwemabhakitiriya. Iri muboka remishonga inorwisa mabhakitiriya inozivikanwa semishonga yesulfa, inoshanda nekudzivisa kukura kwebhakitiriya uye kuberekana kwaro. Sulfadimidine inokanganisa kugadzirwa kwefolic acid mumabhakitiriya, chinhu chakakosha pakurarama kwawo, zvichiita kuti hutachiona hushande zvakanaka pakurwisa mabhakitiriya akasiyana-siyana ane gram-positive negram-negative.
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Sulfacetamide sodium munyu CAS:6209-17-2
Sulfacetamide sodium salt imushonga unonyungudika mumvura wesulfacetamide, mushonga unorwisa mabhakitiriya wesulfonamide unoshandiswa zvakanyanya mukurapa hutachiona hweganda nemaziso. Munyu uyu unowedzera kunyungudika uye kugadzikana kwesulfacetamide, zvichiita kuti ive yakakodzera kushandiswa mumishonga yakasiyana-siyana. Sulfacetamide sodium salt inoshanda nekudzivirira kukura kwebhakitiriya, kunyanya iyo inokonzera zvirwere zvakaita seacne vulgaris, seborrheic dermatitis, uye hutachiona hwemaziso senge conjunctivitis. Inokanganisa kugadzirwa kwefolate yebhakitiriya, ichinyatso tarisa mabhakitiriya akawanda egram-positive negram-negative.
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Streptomycin sulfate CAS:3810-74-0
Streptomycin sulfate mushonga unorwisa mabhakitiriya uri muboka reaminoglycoside. Unobva kubhakitiriya rinonzi Streptomyces griseus uye unoshandiswa zvakanyanya kurapa hutachiona hwehutachiona. Streptomycin sulfate inoshanda nekudzivisa kugadzirwa kwemapuroteni ebhakitiriya, nokudaro ichiuraya mabhakitiriya anonyanya kubatwa nehutachiona. Inowanzo nyorerwa kurapa TB, denda, tularemia, nezvimwe zvirwere zvinokonzerwa nemabhakitiriya anonyanya kubatwa nehutachiona. Streptomycin sulfate inowanzo kuwanikwa muchimiro chejekiseni uye inopihwa kungave ne intramuscularly kana ne intravenously pasi pekutarisirwa kwachiremba.
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Sulfamethoxazole sodium munyu CAS:4563-84-2
Munyu weSulfamethoxazole sodium unobva musulfamethoxazole, mushonga unorwisa mabhakitiriya unoshandiswa mukurapa hutachiona hwemabhakitiriya. Munyu uyu unowedzera kunyungudika uye kugadzikana kwesulfamethoxazole, zvichiita kuti ikodzere mishonga yakasiyana-siyana. Munyu weSulfamethoxazole sodium une simba rekudzivirira kuumbwa kwefolic acid mumabhakitiriya, chinhu chakakosha pakukura kwawo uye kuberekana kwawo. Unoshanda pakurwisa mabhakitiriya akasiyana-siyana ane gram-positive ne gram-negative.
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Sulfamethoxazole CAS:723-46-6
Sulfamethoxazole mushonga unorwisa mabhakitiriya unoshandiswa pamwe chete netrimethoprim kugadzira mushonga une simba unorwisa mabhakitiriya unozivikanwa se co-trimoxazole kana trimethoprim-sulfamethoxazole (TMP-SMX). Iri muboka remishonga inorwisa mabhakitiriya inozivikanwa se sulfa drugs, iyo inodzivirira kukura kwebhakitiriya nekuvhiringidza kugadzirwa kwe folic acid. Sulfamethoxazole inonyanya kurwisa dihydropteroate synthase, enzyme inobatsira mukugadzirwa kwe folate, nokudaro ichiita basa re bacteriostatic kurwisa mabhakitiriya akawanda ane gram-positive ne gram-negative.
