Bhandi neMugwagwa: Kushandira Pamwe, Kuwirirana uye Kukunda-Kukunda
zvigadzirwa

Zvigadzirwa

Venlafaxine CAS:93413-69-5

Venlafaxine mushonga wekudzora kushushikana uri muboka re serotonin ne norepinephrine reuptake inhibitor (SNRI). Mushonga uyu wakagadzirwa kekutanga naWyeth mu19Chemicalbook93 uye ikozvino uri kutengeswa nePfizer. Mushonga uyu unotenderwa kurapa chirwere chikuru chekushungurudzika (MDD), chirwere chekushushikana chakapararira (GAD), uye kushungurudzika kunokonzerwa nekuzvidya mwoyo.


Ruzivo rweChigadzirwa

Matagi eChigadzirwa

Kushandiswa uye Mhedzisiro

Venlafaxine inogona kudzivirira kudzokororwa kweNA ne5-HT, uye zvakare kudzivirira kudzokororwa kwedopamine zvishoma. Kudziviswa kwe cholinergic receptors mu in vitro, histamine receptors α Ma receptors ese ari maviri haana hukama. Kunyudzwa kwemudumbu kwakanaka, uye Chemicalbook inogadziriswa ne cytochrome P45011D6 muchiropa uye inoburitswa nemuweti. T1/2 yemametabolites makuru anoshanda inotangira pamaawa mashanu kusvika gumi nerimwe. Mushure memavhiki matatu, huwandu hwakagadzikana hwakasvika. Yakashandiswa kurapa kushungurudzika.

Muenzaniso weChigadzirwa

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Kurongedza Chigadzirwa:

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Mamwe Mashoko:

Kuumbwa C17H27NO2
Kuyedza 99%
Chitarisiko Upfu hwekristalline chena
Nhamba yeCAS 93413-69-5
Kurongedza 25KG
Hupenyu hweSherufu makore maviri
Kuchengetera Chengeta munzvimbo inotonhorera uye yakaoma
Chitupa ISO.

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