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Ethyl oxalyl monochloride CAS:4755-77-5
Ethyl oxalyl monochloride chinhu chakakosha cheorganic chinoratidzwa neboka re ethyl rakabatana ne oxalyl moiety, iro rine mapoka maviri e carbonyl uye atomu imwe chete ye chlorine. Ne molecular formula C5H7ClO3, chinhu ichi chinozivikanwa zvakanyanya sechikamu chakakosha mukugadzirwa kwe organic, kunyanya mumaindasitiri emishonga ne agrochemicals. Kushanda kwaro kwakasiyana kunobva mukushanda kwaro kwe oxalyl ne chlorinated, zvichibvumira kuti iite shanduko dzakasiyana dzemakemikari. Vaongorori vakaongorora ethyl oxalyl monochloride kuti vaone mashandisirwo ayo mukugadzira mamorekuru akaomarara ane mabasa akasiyana-siyana e biological.
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DL-4-Chlorophenylglycine CAS:6212-33-5
DL-4-Chlorophenylglycine ikemikari yakawana kufarira kukuru muminda yemishonga uye pharmacology. Semushonga unobva kuglycine, ine boka re chlorophenyl, iro rinosimudzira hunhu hwayo hwekubatana uye mashandiro ehupenyu. Kemikari iyi yakaongororwa nekuda kwekushandiswa kwayo mukurapa zvirwere zvakasiyana-siyana zvetsinga, kunyanya nekugadzirisa ma glutamate receptors. Maumbirwo akasiyana eDL-4-Chlorophenylglycine anoibvumirawo kushanda semupikisi kana agonist zvichienderana nenzvimbo yayo, zvichiita kuti ive mukana wekutsvaga mishonga ye neuropharmacological. Kugadzirwa kwayo uye hunhu hwayo zvinoramba zviri nzvimbo dzekuferefeta.
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DRONEDARONE HYDROCHLORIDE CAS:141625-93-6
Dronedarone hydrochloride mushonga unoderedza kusagadzikana kwepfungwa unoshandiswa zvakanyanya mukurapa kusagadzikana kwepfungwa uye kuputika kweropa. Unobva mu amiodarone, wakagadzirwa kuti upe mabhenefiti akafanana ekurapa uku uchideredza mimwe migumisiro yakaipa inokonzerwa ne amiodarone, kunyanya chepfu ye thyroid nemapapu. Dronedarone inoshanda nekuwedzera simba rekuita uye nguva yekuramba kushanda munyama dzemwoyo, ichidzikamisa kumhanya kwemoyo, uye ichideredza njodzi yekuiswa muchipatara nekuda kwezviitiko zvemwoyo. Yakatenderwa kushandiswa mukiriniki munyika dzakasiyana-siyana, dronedarone inomiririra kufambira mberi kukuru mukutarisira mishonga yekushaya simba kwepfungwa.
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valproic acid CAS:99-66-1
Valproic acid, inozivikanwawo se2-propylpentanoic acid, mushonga unoshandiswa zvakanyanya wekurwisa pfari uye kugadzirisa mafungiro, unonyanya kunyorerwa kurapa pfari nebipolar disorder. Yakawanikwa muma1960, inoshanda nekuwedzera huwandu hwegamma-aminobutyric acid (GABA) muuropi, neurotransmitter inokosha inobatsira kudzora kufambisa kwetsinga. Valproic acid yawana kuzivikanwa kwete chete nekuda kwekushanda kwayo mukugadzirisa pfari asiwo nekuda kwebasa rayo mukudzivirira migraines nekurapa mamwe mamiriro epfungwa. Kuonekwa kwayo kwakanaka kwemishonga kunoita kuti ive mushonga unokosha mukurapa tsinga nepfungwa.
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Sodium Valproate CAS:1069-66-5
Sodium valproate, munyu we sodium uri mu valproic acid, mushonga unoderedza pfari uye unodzikamisa mafungiro unoshandiswa zvakanyanya mukurapa pfari ne bipolar disorder. Unoshanda nekuwedzera huwandu hwe gamma-aminobutyric acid (GABA) muuropi, neurotransmitter inoita basa rakakosha mukuderedza kushamisika kwetsinga dzeropa. Yakatenderwa mukupera kwezana remakore rechi20, sodium valproate inozivikanwa nekushanda kwayo mumhando dzakasiyana dzepfari uye inoshandiswawo mukudzivirira migraine. Kuonekwa kwayo kwakanaka kwemishonga kwakaita kuti ive sarudzo yakakosha yekurapa mu neurology ne psychiatry.
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ETHYL 5-AMINOBENZOFURAN-2-CARBOXYLATE CAS:174775-48-5
Ethyl 5-aminobenzofuran-2-carboxylate ikemikari inowanikwa muboka rezvigadzirwa zvebenzofuran, izvo zvakakosha mukemikari yekurapa nekuda kwemabasa avo akasiyana-siyana ehupenyu. Iyi kemikari ine boka rinoshanda re ethyl ester uye inotsiva amino parin'i yebenzofuran, zvichiita kuti ive chinhu chinoshanda pakugadzira mamorekuru anoshanda. Ethyl 5-aminobenzofuran-2-carboxylate yakwezva kutariswa mukutsvaga mishonga nekuda kwekushandiswa kwayo mukugadzira mishonga mitsva yekurapa, kunyanya munzvimbo dzakadai sekurapa kwekudzivirira kuzvimba, kunyaradza marwadzo, kana kuuraya utachiona, nekuda kwehunhu hwayo hwechimiro hunowanikwa nebenzofuran scaffold.
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Diethyl benzylmalonate CAS:607-81-8
Diethyl benzylmalonate chinhu chakakosha cheorganic chinoshandiswa zvakanyanya mumakemikari ekugadzira, kunyanya mukugadzira mishonga yakasiyana-siyana uye agrochemicals. Ichi chinobva kumalonic acid chine mapoka maviri e ethyl ester uye benzyl substituent, iyo inowedzera reactivity yayo mu nucleophilic substitution reactions. Diethyl benzylmalonate inoshanda sechivako chinoshanduka-shanduka mukugadzirwa kwemamorekuru anoshanda mu biologically, kusanganisira zvinhu zvakakosha mukugadzirwa kwemishonga. Maumbirwo ayo akasiyana uye hunhu hwayo hunoita kuti ive chinhu chakakosha mumakemikari ekurapa, zvichibvumira ma chemistry kutsvaga nzira dzakasiyana-siyana dzekugadzira mishonga mitsva.
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Indazole CAS:271-44-3
Indazole imusanganiswa wezvinonhuwira webicyclic une mhete yepyrazole ine nhengo shanu yakabatana nemhete yebenzene ine nhengo nhanhatu. Maumbirwo aya anozivikanwa nekuda kwemabasa ayo akasiyana-siyana ehupenyu uye kushandiswa kwayo mumakemikari ekurapa. Indazole nezvimwe zvinobva mairi zvakawana kutariswa kukuru nekuda kwekubatanidzwa kwavo muzvinhu zvakasiyana-siyana zvemishonga, zvakaita sekudzivirira kuzvimba, kurwisa kenza, uye kuuraya utachiona. Musanganiswa uyu unoshanda senzvimbo yakakosha mukugadzirwa kwemishonga, kunyanya mukugadzirwa kwemishonga mitsva inotarisa zvirwere zvakawanda. Tsvagiridzo iri kuenderera mberi ichienderera mberi nekutsvaga nzira dzekugadzira uye mhedzisiro yehupenyu ine chekuita neindazole.
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ETHYL 5-NITROBENZOURAN-2-CARBOXYLATE CAS:69604-00-8
Ethyl 5-nitrobenzofuran-2-carboxylate chinhu chakakosha muchikamu chemakemikari echisikigo, kunyanya mukati memakemikari eheterocyclic. Sechinhu chinotorwa sebenzofuran chine nitro-substituted, ine hunhu hwakasiyana hwemakemikari uye mabasa ehupenyu anoita kuti ive chinangwa chinokwezva chekutsvagisa kwemishonga. Kuvapo kweboka re nitro kunowedzera reactivity yayo, zvichibvumira kushandiswa kunogona kuitika mukugadzirwa kwemishonga mitsva. Ethyl 5-nitrobenzofuran-2-carboxylate yakwezva kutariswa kwekushandiswa kwayo mukugadzira mishonga inorwisa kuzvimba, inorwisa utachiona, uye inorwisa kenza, ichiratidza kukosha kwayo mukusimudzira nzira dzekurapa dzemakemikari uye kuwana mishonga.
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4-Bromophenylacetone CAS: 6186-22-7
4-Bromophenylacetone iketone inonhuhwirira inozivikanwa nechinhu chinotsiva bromine pa phenyl ring, pamwe chete neboka re acetone rinoshanda. Musanganiswa uyu wakwezva kutariswa mukugadzirwa kwe organic nekuda kwekushanda kwaro kwakasiyana-siyana sechivako mukugadzirwa kwemamorekuru akaomarara, kusanganisira mishonga uye agrochemicals. Kuvapo kweatomu ye bromine kunowedzera hunhu hwayo hwe electrophilic, zvichiita kuti maitiro akasiyana-siyana ashande. Pamusoro pezvo, 4-bromophenylacetone yakaratidza mabasa anogona kuitika muhupenyu, zvichiita kuti ive chinhu chinodiwa mu chemistry yekurapa kuti iwedzere kuongororwa uye kushandiswa mukuwana mishonga.
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4-Hydroxyphenylacetone CAS:770-39-8
4-Hydroxyphenylacetone iketone inonhuhwirira ine boka rehydroxyl rakabatana nephenyl ring uye chikamu cheacetone. Mushonga uyu unozivikanwa nekuda kwekushandiswa kwawo kwakasiyana-siyana mukugadzirwa kweorganic uye chemistry yekurapa. Inoshanda sechikamu chakakosha mukugadzirira mishonga yakasiyana-siyana, agrochemicals, uye makemikari akanaka. Kuvapo kweboka rehydroxy kunowedzera reactivity yayo uye kunobvumira zvimwe shanduko, zvichiita kuti ive nzvimbo inokosha yekugadzira mishonga. Tsvagiridzo mu4-hydroxyphenylacetone yakaratidza mabasa ayo ehupenyu, anosanganisira antioxidant uye anti-inflammatory properties, izvo zvinobatsira pakukosha kwayo muzvidzidzo zvemishonga.
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3-(4-Chlorbutyl)-1H-indol-5-carbonitril CAS:143612-79-7
3-(4-Chlorobutyl)-1H-indol-5-carbonitrile imhando yemusanganiswa weindole unozivikanwa nemusanganiswa wakasiyana wemapoka anoshanda eindole nenitrile, pamwe chete ne chlorobutyl side chain. Musanganiswa uyu wakakurumbira mumunda wekemikari yemishonga nekuda kwemabasa ayo ehupenyu, ayo anogona kusanganisira kuuraya utachiona, kurwisa kuzvimba, uye kurwisa kenza. Musanganiswa weindole unoshanda semusana wekugadzira mishonga, nepo kuvapo kweboka rechlorobutyl kuchiwedzera lipophilicity yayo, zvichigona kuvandudza kuwanikwa kwemishonga. Tsvagiridzo iri kuenderera mberi ine chinangwa chekuongorora mashandisirwo ekurapa uye nzira dzekuita zvine chekuita nemusanganiswa uyu.
