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Clascoterone CAS:19608-29-8 Mugadziri weMugadziri
Clascoterone mushonga unodzivirira androgen receptor uri kugadzirwa sekirimu uye mushonga wepamusoro neCassiopea (kambani inosanganisa Cosmo Pharmaceuticals) yekurapa zvirwere zveganda zvinotsamira pa androgen, zvinosanganisira androgenetic alopecia uye acne vulgaris. Kunyangwe nzira chaiyo yekushanda kwe clascoterone pakurapa acne vulgaris isingazivikanwe, mushonga uyu unofungidzirwa kuti unokwikwidzana ne androgen dihydrotestosterone pakusunga kune androgen receptors mu sebaceous gland uye bvudzi follicles kuderedza zviratidzo zvinodiwa pakukura kwe acne.
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Pitavastatin CAS:147511-69-1 Mugadziri weMugadziri
Pitavastatin inodzivirira HMG-CoA reductase iyo inokonzeresa danho rekutanga rekugadzirwa kwecholesterol. Inoita seisina hwema uye ichena kusvika pahupfu hweyero yakachenuruka. Inobatsira nekuderedza huwandu hwezvimwe zvinhu zvine mafuta zvakaita secholesterol mumuviri. Nokudaro, inonyanya kuratidzwa pakurapa hypercholesterolaemia uye kudzivirira zvirwere zvemwoyo. Haingogone kuderedza cholesterol yakakwira chete uye triglyceride mune vamwe varwere, asiwo inogona kuwedzera huwandu hwe high density lipoprotein (HDL), iyo "cholesterol" yakanaka. Inofanirwa kupihwa pamwe chete nekudya kwakakodzera.
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Teduglutide CAS:197922-42-2 Mugadziri weTeduglutide
Teduglutide (inozivikanwawo seALX-0600) imhando yeGLP-2 iyo glycine yakatsiviwa nealanine panzvimbo yechipiri kubva kuN-terminus, nokudaro ichipa simba rekudzivirira kuora kwemasero neDPP-4. Teduglutide ine hukama hwakafanana, simba reagonist, uye kushanda kweagonist seGLP-2 mukuyedzwa neGLP-2 receptor yemakonzo. Kupihwa kweteduglutide kumakonzo kwakawedzera huremu hwematumbu madiki uye kuwedzera kwehurefu hweintestinal villi. Teduglutide yakagadzirwa ne solid-phase peptide synthesis.
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Malic Acid CAS: 6915-15-7 Mugadziri Mutengesi
Malic acid i2-hydroxydicarboxylic acid iri succinic acid umo imwe yemahydrogens akabatana nekabhoni inotsiviwa neboka rehydroxy. Ine basa rekutonga acidity yechikafu uye metabolite inokosha. I2-hydroxydicarboxylic acid uye C4-dicarboxylic acid. Inobva kusuccinic acid. Iconjugate acid ye malate(2-) uye malate.
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Gabapentin CAS: 60142-96-3 Mugadziri weMugadziri
Gabapentin ineurotransmitter huru inodzivirira inoshanda nekusunga kuma GABA receptors ari mumuzongoza. Gabapentin imhando ye γ-aminobutyric acid (GABA) inoshanda semushonga wekudzivirira marwadzo ane mhedzisiro yakaratidzwa mukurwadziwa kwakasiyana-siyana kweuropi senge Complex Regional Pain Syndrome type one (CRPS 1).
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Paracetamol CAS:103-90-2 Mugadziri weMugadziri
Paracetamol inhengo yeboka remaphenols iro riri 4-aminophenol umo rimwe remahydrogens akabatana neboka remaamino rakatsiviwa neboka reacetyl. Rine basa rekuita se cyclooxygenase 2 inhibitor, cyclooxygenase 1 inhibitor, non-narcotic analgesic, antipyretic, non-steroidal anti-inflammatory drug, cyclooxygenase 3 inhibitor, xenobiotic, Environmental contaminant, human blood serum metabolite, hepatotoxic agent, ferroptosis inducer uye geroprotector. Inhengo yephenols uye nhengo yeacetamides. Rinoshanda pamwe chete ne4-aminophenol.
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Aspartate Calcium CAS:10389-09-0 Mugadziri weMugadziri
Karusiyamu yeAspartatendeimwe yemaminerari akawanda mumuviri uye chinhu chakakosha muhupenyu hwedu. Pasina iyo, vanhu havangagoni kuchengetedza mapfupa nemazino akasimba. Inenge 99% yecalcium mumuviri inochengetwa munzvimbo idzi mbiri. Pamusoro pezvo, calcium inobatsira moyo, tsinga, tsandanyama nedzimwe nzira dzemuviri kushanda zvakanaka. Ine chimiro chakasimba chemakemikari, inonyunguduka zvakanaka mumvura uye inonyunguduka zvakanyanya. Ndiyo yechizvarwa chitsva che calcium nutritional fortifier.
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L-Carnitine L-Tartrate CAS:36687-82-8 Mugadziri wezvigadzirwa
L-carnitine chinhu chinogadzirwa neamino acid chinoshandiswa sekuwedzera uremu. L-carnitine-L-tartrate (LCLT) munyu weL-carnitine une tartaric acid. LCLT ine mabasa ekudzivirira chemo uye antioxidant..
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Miconazole CAS:22916-47-8 Mugadziri weMugadziri
Miconazole (Monistat) mushonga wemishonga inodzivirira fungus weimidazole unoshandiswa pakurapa hutachiona hweganda neganda remukati. Utachiona hweCandida, hwakadai se vaginitis, haunyanyi kunyorova kubva paganda kana pamusoro peganda remukati. Kutsamwiswa kweganda neganda remukati kunogona kuitika kana ukashandiswa paganda; misoro, urticaria, uye kurwadziwa mudumbu zvakashumwa nekurapwa kwe vaginitis.
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Pyrroloquinoline Quinone Disodium Munyu CAS:122628-50-6
Munyu wePyrroloquinoline quinone disodium imusanganiswa wequinone unonyungudika mumvura une simba guru rekudzivirira muviri. Chigadzirwa ichi ipfu ine ruvara rutsvuku-ruvara rwebrown. Yakaparadzaniswa nemarudzi emabhakitiriya emethylotrophic nematishu emhuka dzinoyamwisa. Ichi chikafu chakakosha chakakosha kune mhuka dzinoyamwisa, chichiita basa rakakosha mukusimudzira mashandiro emuviri.
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Citrulline CAS: 372-75-8 Mugadziri weMugadziri
Citrulline ndiyo L-enantiomer ye citrulline. Ine basa rekudzivirira EC 1.14.13.39 (nitric oxide synthase), inodzivirira, ine nutraceutical, ine micronutrient, ine human metabolite, ine Escherichia coli metabolite, ine Saccharomyces cerevisiae metabolite uye ine mbeva metabolite. Ino enantiomer ye D-citrulline. Ino tautomer ye L-citrulline zwitterion.
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L-Arginine Alpha-Ketoglutarate (2:1) Dihydrate CAS:5256-76-8
L-Arginine Alpha-Ketoglutarate (2: 1) Dihydratemushonga wemishonga uri muboka remishonga inoshandiswa kurapa hyperlipidemia. Maumbirwo emushonga uyu ane mamorekuru maviri earginine akabatanidzwa neatomu yeokisijeni. Ikristaro yakasimba ine avhareji yedhayamita yezvikamu zve 0.3 μm uye kugoverwa kwezvikamu zvezvikamu kunobva pa 0.05 kusvika 1.5 μm.
